2017

• Fredrik, Bysting; Bugge, Steffen; Sundby, Eirik; Hoff, Bård Helge. (2017) Investigation of Heck coupling on 6-bromo[2,3-d]thienopyrimidines for construction of new EGFR inhibitor lead structures. RSC Advances. vol. 7.
• Haghdani, Shokouh; Hoff, Bård Helge; Koch, Henrik; Åstrand, Per-Olof. (2017) Solvent Effects on Optical Rotation: On the Balance between Hydrogen Bonding and Shifts in Dihedral Angles. Journal of Physical Chemistry A. vol. 121 (5).
• Petrovic, Voin; Olaisen, Camilla; Sharma, Animesh; Nepal, Anala; Bugge, Steffen; Sundby, Eirik; Hoff, Bård Helge; Slupphaug, Geir; Otterlei, Marit. (2017) On-column trypsinization allows for re-use of matrix in modified multiplexed inhibitor beads assay. Analytical Biochemistry. vol. 523.

2016

• Bugge, Steffen; Buene, Audun Formo; Jurisch-Yaksi, Nathalie; Moen, Ingri Ullestad; Skjønsfjell, Ellen Martine; Sundby, Eirik; Hoff, Bård Helge. (2016) Extended structure-activity study of thienopyrimidine-based EGFR inhibitors with evaluation of drug-like properties. European Journal of Medicinal Chemistry. vol. 107.
• Haghdani, Shokouh; Hoff, Bård Helge; Koch, Henrik; Åstrand, Per-Olof. (2016) Optical Rotation Calculations for Fluorinated Alcohols, Amines, Amides, and Esters. Journal of Physical Chemistry A. vol. 120 (40).
• Han, Jin; Henriksen, Silje; Nørsett, Kristin Gabestad; Sundby, Eirik; Hoff, Bård Helge. (2016) Balancing potency, metabolic stability and permeability in pyrrolopyrimidine-based EGFR inhibitors. European Journal of Medicinal Chemistry. vol. 124.
• Han, Jin; Kaspersen, Svein Jacob; Nervik, Sondre; Nørsett, Kristin; Sundby, Eirik; Hoff, Bård Helge. (2016) Chiral 6-aryl-furo[2,3-d]pyrimidin-4-amines as EGFR inhibitors. European Journal of Medicinal Chemistry. vol. 119.

2015

• Bugge, Steffen; Moen, Ingri Ullestad; Sylte, Kent-Ove Kragseth; Sundby, Eirik; Hoff, Bård Helge. (2015) Truncated structures used in search for new lead compounds and in a retrospective analysis of thienopyrimidine-based EGFR inhibitors. European Journal of Medicinal Chemistry. vol. 94.
• Gulbrandsen, Tore Aarhus; Johnsen, Ingvild Andersen; Opedal, Mihaela Tanase; Toven, Kai; Øyaas, Karin; Pranovich, Andrey; Mikkola, Jyri-Pekka; Hoff, Bård Helge. (2015) Extracting hemicelluloses from softwood and bagasse as oligosaccharides using pure water and microwave heating. Cellulose Chemistry and Technology. vol. 49 (2).
• Karlsen, Morten; Liu, Huiling; Johansen, Jon Eigill; Hoff, Bård Helge. (2015) Economical Synthesis of 13C-Labeled Opiates, Cocaine Derivatives and Selected Urinary Metabolites by Derivatization of the Natural Products. Molecules. vol. 20 (4).
• Sundby, Eirik; Han, Jin; Kaspersen, Svein Jacob; Hoff, Bård Helge. (2015) In vitro baselining of new pyrrolopyrimidine EGFR-TK inhibitors with Erlotinib. European Journal of Pharmaceutical Sciences. vol. 80.

2014

• Bugge, Steffen; Kaspersen, Svein Jacob; Larsen, Synne; Nonstad, Unni; Bjørkøy, Geir; Sundby, Eirik; Hoff, Bård Helge. (2014) Structure-activity study leading to identification of a highly active thienopyrimidine based EGFR inhibitor. European Journal of Medicinal Chemistry. vol. 75.
• Bugge, Steffen; Skjønsfjell, Ellen Martine; Willumsen, Fredrik Bysting; Sundby, Eirik; Hoff, Bård Helge. (2014) Improved and Scalable Preparation of 6-Bromo-4-Chlorothieno[2,3-d]Pyrimidine. Chemistry of Heterocyclic Compounds. vol. 50 (8).
• Karlsen, Morten; Liu, Huiling; Berg, Thomas; Johansen, Jon Eigill; Hoff, Bård Helge. (2014) Synthesis of [13C6]-labelled phenethylamine derivatives for drug quantification in biological samples. Journal of labelled compounds & radiopharmaceuticals. vol. 57 (5).
• Karlsen, Morten; Liu, Huiling; Johansen, Jon Eigill; Hoff, Bård Helge. (2014) Synthesis of [13C4]-labeled ∆9-tetrahydrocannabinol and 11-nor-9-carboxy-∆9-tetrahydrocannabinol as internal standards for reducing ion supressing/alteration effects in LC/MS-MS quantification. Molecules. vol. 19 (9).
• Kaspersen, Svein Jacob; Han, Jin; Nørsett, Kristin; Rydså, Line; Kjøbli, Eli; Bugge, Steffen; Bjørkøy, Geir; Sundby, Eirik; Hoff, Bård Helge. (2014) Identification of new 4-N-substituted 6-aryl-7H-pyrrolo[2,3-d]pyrimidine-4- amines as highly potent EGFR-TK inhibitors with Src-family activity. European Journal of Pharmaceutical Sciences. vol. 59 (1).

2013

• Han, Jin; Sundby, Eirik; Hoff, Bård Helge. (2013) Solvent selection in synthesis of 4-(1-arylfluoroethoxy)quinazolines and thienopyrimidines. Journal of fluorine chemistry. vol. 153.
• Hoff, Bård Helge; Sundby, Eirik. (2013) Preparation of pharmaceutical important fluorinated 1-arylethanols using isolated enzymes. Bioorganic chemistry (Print). vol. 51C.
• Rodionova, Galina; Hoff, Bård Helge; Lenes, Marianne; Eriksen, Øyvind; Gregersen, Øyvind Weiby. (2013) Gas-phase esterification of microfibrillated cellulose (MFC) films. Cellulose (London). vol. 20 (3).
• Thvedt, Thor Håkon Krane; Kaasa, Kristin; Sundby, Eirik; Charnock, Colin; Hoff, Bård Helge. (2013) Chiral N-benzyl-N-methyl-1-(naphthalen-1-yl)ethanamines and their in vitro antifungal activity against Cryptococcus neoformans, Trichophyton mentagrophytes and Trichophyton rubrum. European Journal of Medicinal Chemistry. vol. 68.

2012

• Bugge, Steffen; Kaspersen, Svein Jacob; Sundby, Eirik; Hoff, Bård Helge. (2012) Route selection in the synthesis of C-4 and C-6 substituted thienopyrimidines. Tetrahedron. vol. 68 (45).
• Esmurziev, Aslan; Reimers, Arne; Andreassen, Trygve; Simic, Nebojsa; Sundby, Eirik; Hoff, Bård Helge. (2012) Benzoylated uronic Acid building blocks and synthesis of N-uronate conjugates of lamotrigine. Molecules. vol. 17 (1).
• Kaspersen, Svein Jacob; Sundby, Eirik; Charnock, Colin; Hoff, Bård Helge. (2012) Activity of 6-aryl-pyrrolo[2,3-d]pyrimidine-4-amines to Tetrahymena. Bioorganic chemistry (Print). vol. 44.

2011

• Kaspersen, Svein Jacob; Sørum, Christopher; Willassen, Veronica; Fuglseth, Erik; Kjøbli, Eli; Bjørkøy, Geir; Sundby, Eirik; Hoff, Bård Helge. (2011) Synthesis and in vitro EGFR (ErbB1) tyrosine kinase inhibitory activity of 4-N-substituted 6-aryl-7H-pyrrolo[2,3-d]pyrimidine-4-amines. European Journal of Medicinal Chemistry. vol. 46 (12).
• Slungård, Sigrid Volden; Krakeli, Tor-Arne; Thvedt, Thor Håkon Krane; Fuglseth, Erik; Sundby, Eirik; Hoff, Bård Helge. (2011) Investigation into the enantioselection mechanism of ruthenium-arene-diamine transfer hydrogenation catalysts using fluorinated substrates. Tetrahedron. vol. 67 (31).
• Thvedt, Thor Håkon Krane; Kristensen, Tor Erik Holt; Sundby, Eirik; Hansen, Tore; Hoff, Bård Helge. (2011) Enantioselectivity, swelling and stability of 4-hydroxyprolinol containing acrylic polymer beads in the asymmetric reduction of ketones. Tetrahedron: asymmetry. vol. 22 (24).

2010

• Esmurziev, Aslan; Simic, Nebojsa; Hoff, Bård Helge; Sundby, Eirik. (2010) Synthesis and Structure Elucidation of Benzoylated Deoxyfluoropyranosides. Journal of carbohydrate chemistry. vol. 29 (7).
• Lystvet, Sina Maria; Hoff, Bård Helge; Anthonsen, Thorleif; Jacobsen, Elisabeth Egholm. (2010) Chemoenzymatic synthesis of enantiopure 1-phenyl-2-haloethanols and their esters. Biocatalysis and Biotransformation. vol. 28 (4).
• Sørum, Christopher; Simic, Nebojsa; Sundby, Eirik; Hoff, Bård Helge. (2010) 1H,13C and 19F NMR data of N-substituted 6-(4-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amines in DMSO-d6. Magnetic Resonance in Chemistry. vol. 48 (3).
• Thvedt, Thor Håkon Krane; Fuglseth, Erik; Sundby, Eirik; Hoff, Bård Helge. (2010) Enantioenriched 1-aryl-2-fluoroethylamines. Efficient lipase-catalysed resolution and limitations to the Mitsunobu inversion protocol. Tetrahedron. vol. 66 (34).

2009

• Esmurziev, Aslan; Simic, N.; Sundby, Eirik; Hoff, Bård Helge. (2009) H-1 and C-13 NMR data of methyl tetra-O-benzoyl-D-pyranosides in acetone-d(6). Magnetic Resonance in Chemistry. vol. 47 (5).
• Esmurziev, Aslan; Simic, Nebojsa; Sundby, Eirik; Hoff, Bård Helge. (2009) 1H and 13C NMR data of methyl tetra-O-benzoyl-D-pyranosides in acetone-d6. Magnetic Resonance in Chemistry. vol. 47 (5).
• Esmurziev, Aslan; Sundby, Eirik; Hoff, Bård Helge. (2009) Regioselective C-6 Hydrolysis of Methyl O-Benzoyl-pyranosides Catalysed by Candida Rugosa Lipase. European Journal of Organic Chemistry. vol. 10.
• Esmurziev, Aslan; Sundby, Eirik; Hoff, Bård Helge. (2009) Regioselective C-6 Hydrolysis of Methyl O-Benzoyl-pyranosides Catalysed by Candida Rugosa Lipase. European Journal of Organic Chemistry.
• Fuglseth, Erik; Otterholt, Eli; Høgmoen, Hanne; Høgmoen, Hanne; Sundby, Eirik; Sundby, Eirik; Charnock, Colin; Hoff, Bård Helge. (2009) Chiral derivatives of Butenafine and Terbinafine: synthesis and antifungal activity. Tetrahedron. vol. 65 (47).
• Fuglseth, Erik; Sundby, Eirik; Hoff, Bård Helge. (2009) Ruthenium-catalysed asymmetric transfer hydrogenation of para-substituted alpha-fluoroacetophenones. Journal of fluorine chemistry. vol. 130 (6).
• Fuglseth, Erik; Sundby, Eirik; Hoff, Bård Helge. (2009) Ruthenium-catalysed asymmetric transfer hydrogenation of para-substituted alpha-fluoroacetophenones. Journal of fluorine chemistry. vol. 130 (6).
• Thvedt, Thor Håkon Krane; Fuglseth, Erik; Sundby, Eirik; Hoff, Bård Helge. (2009) Microwave assisted fluorination: an improved method for side chain fluorination of substituted 1-arylethanones. Tetrahedron. vol. 65 (46).

2008

• Esmurziev, Aslan; Hoff, Bård Helge; Sundby, Eirik. (2008) Regioselective enzymatic hydrolysis of tetrabenzoylated hexapyranosides. Biocatalysis in Non-Convential Medium . Moskvas stalig universitet; Moskva. 2008-06-11 - 2008-06-16.
• Fuglseth, Erik; Sundby, Eirik; Bruheim, Per; Hoff, Bård Helge. (2008) Asymmetric reduction using (R)-MeCBS and determination of absolute configuration of para-substituted 2-fluoroarylethanols. Tetrahedron: asymmetry. vol. 19.
• Fuglseth, Erik; Sundby, Eirik; Bruheim, Per; Hoff, Bård Helge. (2008) Asymmetric reduction using (R)-MeCBS and determination of absolute configuration of para-substituted 2-fluoroarylethanols. Tetrahedron: asymmetry. vol. 19 (16).
• Fuglseth, Erik; Thvedt, Thor Håkon Krane; Møll, Maria Førde; Hoff, Bård Helge. (2008) Electrophilic and nucleophilic side chain fluorination of para-substituted acetophenones. Tetrahedron. vol. 64.

2006

• Hoff, Bård Helge; Anthonsen, Thorleif; Fuglseth, Erik. (2006) New chiral building blocks from acetovanillone using lipase A and B from Candida antarctica. Tetrahedron: asymmetry. vol. 17 (8).

2004

• Moen, A. R.; Hoff, B. H.; Hansen, Lars Kr; Anthonsen, T.; Jacobsen, E. E.. (2004) Absolute configurations of monoesters produced by enzyme catalyzed hydrolysis of diethyl 3-hydroxyglutarate. Tetrahedron: asymmetry. vol. 15.

2003

• Jacobsen, Elisabeth Egholm; Hoff, Bård Helge; Moen, Anders Riise; Anthonsen, Thorleif. (2003) Enantioselective enzymatic preparation of chiral glutaric monocarboxylic acids and amides. Journal of Molecular Catalysis B: Enzymatic. vol. 21.

2002

• Sundby, Eirik; Anthonsen, Thorleif; Andersen, Morten Myhre; Hoff, Bård Helge. (2002) Lipase catalysed resolution and microbial reduction for obtaining enantiopure 1-(2-thienyl)alkanols. ARKIVOC.

2001

• Liu, Hui-Ling; Hoff, Bård Helge; Berg, Tom Christian; Anthonsen, Thorleif. (2001) Synthesis of the anti-stroke drug Lubeluzole and its enantiomer. Lipase catalyzed resolution of chiral building block. Chirality. vol. 13.

2000

• Egholm Jacobsen, Elisabeth; Hoff, Bård Helge; Anthonsen, Thorleif. (2000) Enantiopure derivatives of 1,2-alkanediols. Substrate requirements for lipase B from Candida antarctica. Chirality. vol. 12.
• Hoff, Bård; Ljones, Liv; Rønstad, Anja; Anthonsen, Thorleif. (2000) Influence of Substituents on Enantiomeric Ratio in Transesterification of Racemic C-3 Synthons using Lipase B from Candida antarctica. Journal of Molecular Catalysis B: Enzymatic. vol. 8.
• Jacobsen, Elisabeth Egholm; Hoff, Bård Helge; Anthonsen, Thorleif. (2000) Enantiopure derivatives of 1,2-alkanediols: Substrate requirements of lipase B from Candida antarctica. Chirality. vol. 12.
• Liu, Hui Ling; Hoff, Bård Helge; Anthonsen, Thorleif. (2000) Chemoenzymatic synthesis of the antidepressant Duloxetine and its enantiomer. Chirality. vol. 12.
• Liu, Hui-Ling; Hoff, Bård Helge; Anthonsen, Thorleif. (2000) Chemo-enzymatic synthesis of both enantiomers of the non-tricyclic antidepressants Fluoxetine, Nisoxetine and Tomoxetine. Journal of the Chemical Society. Perkin transactions 1.

1999

• Anthonsen, Thorleif; Hoff, Bård Helge. (1999) Gas Chromatographic enantiomer separation of C-3 and C-4 synthons. Combination with enzymatic resolution to determine absolute configuration. Chirality. vol. 11.
• Anthonsen, Thorleif; Hoff, Bård Helge; Hofsløkken, Nini; Skattebøl, Lars; Sundby, Eirik. (1999) Synthesis of 1,3-dithianes and 1,3-dithiolanes. Baker´s yeast reduction and lipase-catalyzed resolution for synthesis of enantiopure derivatives. Acta Chemica Scandinavica. vol. 53.
• Anthonsen, Thorleif; Hoff, Bård Helge; Liu, Hui-Ling; Sundby, Eirik. (1999) Enantiopure chiral building blocks by biocatalysis. Metal and bio-promoted selective organic transformations. COST D12 Workshop . [Mangler data]; Sassari-Porto Conte, Italia, Oktober 1999.
• Berg, Tom Christian; Hoff, Bård Helge; Anthonsen, Thorleif. (1999) Chemo-enzymatic synthesis of the drug Lubeluzole. 7. Nordic Conference on Biocatalysis in Organic Chemistry . [Mangler data]; Teveltunet fjellstue, Norway. 8.-11. April 1999.
• Hoff, Bård Helge; Anthonsen, Thorleif. (1999) Lipase catalyzed resolution of esters of 4-chloro-3-hydroxy butanoic acid. Effect of alkoxy group and solvent on enantiomeric ratio. 7. Nordic Conference on Biocatalysis in Organic Chemistry . [Mangler data]; Teveltunet fjellstue, 8.-11. april 1999.
• Hoff, Bård Helge; Anthonsen, Thorleif. (1999) Lipase catalyzed resolution of esters of 4-chloro-3-hydroxybutanoic acid. Effect of alkoxy group and solvent on enantiomeric ratio. Tetrahedron: asymmetry. vol. 10.
• Jacobsen, Elisabeth Egholm; Hoff, Bård Helge; Anthonsen, Thorleif. (1999) Significance of substrate structure, acyl donor and water activity for E in resolutions of secondary alcohols catalysed by CALB. 7. Nordic Conference on Biocatalysis in Organic Chemistry . [Mangler data]; Teveltunet fjellstue, 8- 11. april 1999. 1999-04-17 - 1999-04-20.
• Anthonsen, Thorleif; Hoff, Bård H.; Hofsløkken, Nini Unn; Skattebøl, Lars; Sundby, Eirik. (1999) Synthesis of 1,3-Dithianes and 1,3-Dithiolanes. Baker's Yeast reduction and Lipase-Catalyzed resolution for synthesis of Enantiopure derivatives. Acta Chemica Scandinavica. vol. 53.

1998

• Hoff, Bård; Anthonsen, Thorleif. (1998) Resolution of Derivatives of 1,2-Propanediol with Lipase B from Candida antarctica. Effect of Substrate Structure, Medium, Water Activity and Acyl on Enantiomeric Ratio. Chemistry and Physics of Lipids. vol. 93 (xx).

1997

• Hoff, Bård; Anthonsen, Henrik; Anthonsen, Thorleif. (1997) Lipase catalysed resolution in organic solvent : the enantiomer ratio strongly depends on the alkyl part of the acyl donor in transesterification with lipase B from Candida antarctica. Organisk kjemisk vintermøte . [Mangler data]; Fefor.

1996

• Anthonsen, H.W.; Hoff, B.H.; Anthonsen, Thorleif. (1996) Calculation of enantiomer ratio and equilibrium constants in biocatalytic ping-pong bi-bi resolutions. Tetrahedron: asymmetry. vol. 7.
• Anthonsen, H.W.; Hoff, B.H.; Anthonsen, Thorleif. (1996) Calculation of enantiomer ratio and equilibrium constants in biocatalytic resolutions : resolution of derivatives of 1,2-propanediol. 11. Organisk kjemisk vintermøte . [Mangler data]; [Mangler data].
• Hoff, B.H.; Anthonsen, H.W.; Anthonsen, Thorleif. (1996) The enantiomer ratio strongly depends on the alkyl part of the acyl donor in transesterification with lipase B from Candida antarctica. Tetrahedron: asymmetry. vol. 7.
• Hoff, B.H.; Waagen, V.; Anthonsen, Thorleif. (1996) Resolution of 1-phenoxy-, 1-phenylmethoxy- and 1-(2-phenylethoxy)-2-propanol and their butanoates by hydrolysis with lipase B from Candida antarctica. Tetrahedron: asymmetry. vol. 7.

1995

• Anthonsen, Henrik Walbye; Hoff, Bård Helge; Anthonsen, Thorleif. (1995) A simple method for calculating enantiomer ratio and equilibrium constants in biocatalytic resolutions. Tetrahedron: asymmetry. vol. 6.